Orforglipron 30 x 3mg tabs
$120.00
Orforglipron (30 x 3mg tabs) is the world’s first oral small-molecule GLP-1 receptor agonist — a major breakthrough that delivers the metabolic power of GLP-1 therapy in a simple daily tablet. No injections. No fasting. No food restrictions. Just measurable weight reduction, sharper appetite control, and improved metabolic markers.
In stock
| Title | Range | Discount |
|---|---|---|
| Bulk Discount OptimaSciences | 3 - 4 | 10% |
| Bulk Discount OptimaSciences | 5 + | 15% |
⚠️ Research Use Only (RUO). Not for human or veterinary use.
Orforglipron is a non-peptide small molecule GLP-1 receptor agonist, formula C48H48F2N10O5, 882.97 g/mol. Being a small molecule rather than a peptide is exactly why it survives the stomach and can be taken as a tablet at all, and its two fluorine atoms are a standard approach to slowing metabolic breakdown.
Supplied as 30 oral tablets of 3 mg each, release specification ≥99% by HPLC. Verified and packed in our Ontario lab. No reconstitution and no bacteriostatic water required. The certificate for your batch is in the photos above.
We do not import Orforglipron 30 x 3mg tabs finished. We buy the raw material and do the purification, verification and pressing ourselves, in Ontario.
Additional information
| Weight | 0.1 kg |
|---|---|
| Dimensions | 15 × 15 × 2 cm |
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Why choose Orforglipron
What it is chosen for.
Oral convenience. Phase 3 trials show weight reduction comparable to leading injectable GLP-1 therapies, without the needles or refrigeration.
Powerful appetite control. Modulates hunger signals and cravings, making calorie control feel effortless.
Metabolic reset. Supports healthier blood sugar, lower waist circumference and improved cardiometabolic markers.
Premium quality. Sourced from trusted suppliers, sealed and purity tested for maximum safety.
The compound
Orforglipron, in short.
Not a peptide at all
The only GLP-1 receptor agonist here that is a small molecule. That is precisely why it survives the stomach and can be taken as a tablet.
Two fluorine atoms
Formula C48H48F2N10O5. Fluorine is a favourite trick of medicinal chemists for slowing metabolic breakdown.
Solved in 2020
Kawai and colleagues published the receptor structure in PNAS, under the code LY3502970.
Finished in Ontario, Canada
Verified and packed in our own lab. Full numbers below.
Specification
What is in the tablet, down to the formula.
The molecule
| Class | Non-peptide small molecule GLP-1 receptor agonist |
| Length | Not a peptide |
| CAS number | 2212020-52-3 |
| Formula | C48H48F2N10O5 |
| Molecular weight | 882.97 g/mol |
| Origin | Fully synthetic |
| First described | PNAS, 2020 |
This product
| Fill weight | 3 mg |
| Form | Oral tablet |
| Purity | ≥99% by HPLC · release spec |
| Identity | Confirmed by mass spectrometry |
| Storage | −20 °C, protected from light |
| Manufactured | Ontario, Canada |
The problem with this market
Every vial said 99% pure. None of them were.
Researchers ordered from six online peptide sellers. Half never arrived at all. Here is what was in the three vials that did.
was actually peptide
was actually peptide
was actually peptide
Endotoxin in all three, and no buyer had any way of knowing. Not one of those sellers published a test.
We publish ours. Raw material arrives in Ontario, we purify, verify, fill and freeze dry it here, and the certificate for the batch you receive is in the photos above with the lab and the test date on it.
Three vials is a small sample and the compound was semaglutide, not the one on this page. It is the only peer reviewed teardown of this market that exists, which is itself the point. Ashraf et al., Journal of Medical Internet Research, 2024, DOI 10.2196/65440.
Why buy it here
Same molecule. Different supply chain.
We make it. We do not resell it.
Raw material in, finished vial out, same facility. Most of this market buys vials already filled and puts a label on them.
The certificate is for the batch in the box.
Not an undated PDF from some other run. Replaced here every time a new batch is released, with the lab and the date on it.
Minus 20 °C until it is packed.
Our own freezer to the moment it ships, then tracked with Canada Post. No customs queue, no week at ambient in transit.
Every row is a fact about how the product is made and handled, and every row is one we can evidence.
Before you order
The practical questions.
When will my order ship, and how does it arrive?
Orders placed before 2pm ET are dispatched within 2 business days. Everything goes tracked with Canada Post. Shipping is free on orders over $200.
What exactly is in the box?
A sealed container holding the count shown on this page. Nothing else is required.
How is it stored before it ships?
Every unit is held at −20 °C in our own lab freezer until the moment it is packed.
Where is this made, and who tests it?
Raw material arrives in Ontario and is purified, verified, filled and freeze dried in our own facility. Every batch is tested before it is released.
Can I see the certificate for the batch I will receive?
It is already on this page, in the product photos. Nothing ships until its certificate is back from the lab, and we swap the photo the moment the batch changes, so what you are looking at is what is in the box.
What is your return policy?
Once a product leaves our freezer we cannot
take it back. A product stored somewhere we cannot
see is one we can no longer vouch for, and we will not put it back into circulation
for someone else. So all sales are final.
The exception is anything that is our fault. If what arrives is damaged, defective
or not what you ordered, send us a photo and we will replace it or refund it. Get in
touch soon after delivery so we can act on it while it is still clear what happened.
What we cannot cover is how the product is handled, stored or used once the box
reaches you, for exactly the same reason we cannot take it back.
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Our lab, Ontario
We didn't import these tablets.
We made them.
Purified, verified and pressed in our own Ontario lab. Not bought finished and relabelled.
See how it was made- Raw material
- Purification
- Verification
- Pressing
- Release